化學_產(chǎn)品搜索_第121頁_醫(yī)化信息網(wǎng)

Tozasertib
Tozasertib (MK-0457; VX-680) is the inhibitor of Aurora-A, -B, -C kinases with Ki values of 0.6, 18, 4.6 nM respectively
2016-01-04 16:13 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

1515.00/50mg
050mg起訂

PIK-75
PIK-75 is a p110 inhibitor with IC50 of 5.8 nM (200-fold more potently than p110), isoform-specific mutants at Ser773, a
2016-01-04 16:11 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

512.00/10mg
010mg起訂

Hesperadin
Hesperadin is a ATP-competitive inhibitor of Aurora B kinase with IC50 of 250 nM.IC50 Value: 250 nMTarget: Aurora Bin vi
2016-01-04 16:09 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

1200.00/5mg
05mg起訂

GW 501516
GW501516(GSK-516; GW1516) is a potent and highly selective PPAR/ agonist, with EC50 of 1 nM, with 1000-fold selectivity
2016-01-04 16:07 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

2175.00/10mg
010mg起訂

b-AP15
b-AP15(NSC687852) is a specific inhibitor of the deubiquitinating enzymes UCHL5 and Usp14 of the 26S proteasome. 公司介
2016-01-04 16:05 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

558.00/5mg
05mg起訂

Decitabine
Decitabine is a potent inhibitor of DNA methyltransferase with IC50 of 438 nM and 4.38 nM in HL-60 and KG1a cells, respe
2016-01-04 16:03 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

651.00/10mg
010mg起訂

ROCK inhibitor
ROCK inhibitor(azaindole 1) is a highly potent inhibitor of human ROCK-1 and ROCK-2 isoenzymes with IC50 values of 0.6 a
2016-01-04 16:01 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

3339.00/5mg
05mg起訂

Flavopiridol (Hydrochloride)
Flavopiridol hydrochloride competes with ATP to inhibit CDKs including CDK1, CDK2, CDK4 and CDK6 with IC50 of ~ 40 nM.
2016-01-04 15:59 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

810.00/10mg
010mg起訂

Volasertib
Volasertib(BI6727) is a highly potent PLK1 inhibitor with an IC50 of 0.87 nM; shows 6- and 65-fold greater selectivity a
2016-01-04 15:57 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

893.00/5mg
05mg起訂

Panobinostat
Panobinostat(LBH-589) is a broad-spectrum HDAC inhibitor; low nanomolar concentrations (IC50=5-20 nM) of LBH589 induced
2015-12-25 17:27 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

651.00/10mg
010mg起訂

TAK-901
TAK-901 is a novel inhibitor of Aurora A/B with IC50 of 21 nM/15 nM. 公司介紹：MedChemExpress(MCE)專注于各種抑制劑、激動
2015-12-25 17:26 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

1265.00/5mg
05mg起訂

CDK-IN-2
CDK-IN-2 is a potent and sepecific CDK inhibitor.公司介紹：MedChemExpress(MCE)專注于各種抑制劑、激動劑、API及化合物庫，
2015-12-25 17:23 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

1256.00/5mg
05mg起訂

VE-821
VE-821 is a potent and selective ATP competitive inhibitor of ATR with Ki/IC50 of 13 nM/26 nM.IC50 Value: 26 nMTarget: A
2015-12-25 17:22 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

744.00/5mg
05mg起訂

Fasudil (Hydrochloride)
Fasudil Hcl(HA-1077; AT-877) is a potent inhibitor of ROCK-II, PKA, PKG, PKC, and MLCK with Ki of 0.33 M, 1.6 M, 1.6 M,
2015-12-25 17:13 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

1252.00/500mg
0500mg起訂

Y-27632
Y-27632 is a selective ROCK1 (p160ROCK) inhibitor with Ki of 140 nM, exhibits 200-fold selectivity over other kinases, i
2015-12-25 17:11 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

874.00/5mg
05mg起訂

ENMD-2076 (Tartrate)
ENMD-2076 tartrate has selective activity against Aurora A and Flt3 with IC50 of 14 nM and 1.86 nM, 25-fold selective fo
2015-12-25 17:08 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

515.00/5mg
05mg起訂

CCT129202
CCT129202 is a Aurora kinase inhibitor with IC50 of 0.0420.022, 0.1980.05, and 0.2270.064 uM for Aurora A, Aurora B, and
2015-12-25 17:06 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

1252.00/5mg
05mg起訂

HMN-214
HMN-214(IVX214) is a potent PLK1 inhibitor an average IC50 of 0.12 M.IC50 Value: 0.12 MTarget: PLK1in vitro: HMN-214 is
2015-12-25 17:04 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

7217.00/50mg
050mg起訂

PHA-680632
PHA-680632 is potent inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 27 nM, 135 nM and 120 nM, respectively.公
2015-12-25 17:02 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]

1252.00/5mg
05mg起訂

Rigosertib (sodium)
Rigosertib sodium (ON-01910 sodium) is a non-ATP-competitive inhibitor of PLK1 with IC50 of 9 nM.公司介紹：MedChemExpres
2015-12-25 17:00 [上海]
上海皓元生物醫(yī)藥科技有限公司 [已核實]